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- A3278 Nonivamide (Capsaicin Analog)1 Citation中文名: 香草壬酰胺Target: TRP ChannelSummary: TRPV1受体激动剂
- A1174 AMG-517Target: TRP ChannelSummary: TRPV1拮抗剂
- A8616 A-674563Target: Cyclin-Dependent Kinases|Akt|GSK-3|ERK|PKC|PKA|RSKSummary: Akt1 / PKA / CDK2的强效选择性抑制剂
- A3943 XMD8-92Target: ERKSummary: BMK1/ERK5抑制剂
- B1055 IcilinTarget: TRP ChannelSummary: TRPM8/ hENaCδ激动剂
- B5839 SU6656Target: Src|Lyn|YES|FynSummary: Src 酪氨酸激酶抑制剂
- A2942 Masitinib (AB1010)中文名: 马赛替尼Target: PDGFR|c-Kit|LynSummary: 酪氨酸激酶抑制剂
- B3492 Bedaquiline中文名: 贝达喹啉Target: ATP synthaseSummary: 抗结核药物
- B1106 VRT752271Target: ERKSummary: ERK1/ERK2 inhibitor
- N1311 Nobiletin中文名: 蜜橘黄素,川陈皮素Target: ERKSummary: ERK抑制剂