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- A1185 BMS-754807Target: Insulin and Insulin-like ReceptorsSummary: 有效的、选择性的IGF-1R和InsR抑制剂
- A8440 GSK1838705ATarget: Insulin and Insulin-like Receptors|ALKSummary: ATP竞争性IGF-IR/IR/ALK抑制剂
- A3608 MK 0893Target: Insulin and Insulin-like Receptors|Glucagon ReceptorsSummary: 胰高血糖素受体/ IGF-1R拮抗剂
- A3744 Quetiapine中文名: 喹硫平Target: AChR|adrenergic receptor|5-HT receptor|Dopamine receptor|Histamine receptorSummary: 多巴胺受体拮抗剂
- A3454 GW39651 CitationTarget: Liver X receptors (LXRs)Summary: 高效选择性HLXRα/hLXRβ激动剂
- A3368 DMAT2 CitationTarget: Pim|CK2|HIPK2|HIPK3Summary: CK2抑制剂
- A8714 SR-9243Target: Liver X receptors (LXRs)Summary: LXR反相激动剂
- B1572 LatrepirdineTarget: Voltage-gated Calcium Channels (CaV)|NMDA receptor|adrenergic receptor|Histamine receptors|GluR|5-HT receptor|dopamine receptors|AMPA receptorSummary: 脑细胞死亡抑制剂
- B1264 LXR-6232 CitationTarget: Liver X receptors (LXRs)Summary: 肝X受体激动剂
- A2249 T0901317Target: Liver X receptors (LXRs)Summary: 肝X受体激动剂