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- A1185 BMS-754807Target: Insulin and Insulin-like ReceptorsSummary: 有效的、选择性的IGF-1R和InsR抑制剂
- A8440 GSK1838705ATarget: Insulin and Insulin-like Receptors|ALKSummary: ATP竞争性IGF-IR/IR/ALK抑制剂
- A4424 SID 26681509Target: CathepsinsSummary: 人组织蛋白酶L抑制剂
- A8174 Cathepsin G Inhibitor ITarget: CathepsinsSummary: Cathepsin G抑制剂
- A1926 CA 0742 CitationTarget: CathepsinsSummary: Cathepsin B抑制剂
- A3608 MK 0893Target: Insulin and Insulin-like Receptors|Glucagon ReceptorsSummary: 胰高血糖素受体/ IGF-1R拮抗剂
- A8239 CA-074 Me7 CitationTarget: CathepsinsSummary: Cathepsin B抑制剂
- A2571 Pepstatin A1 Citation中文名: 抑肽素Target: Cathepsins|Renin|HIV proteases|PepsinsSummary: 天冬氨酸蛋白酶抑制剂
- A3284 Cathepsin S inhibitor1 CitationTarget: CathepsinsSummary: 抑制MHCII抗原呈递
- B5437 Decanoyl-RVKR-CMKTarget: Subtilisin/Kex2p-like proprotein convertaseSummary: 枯草杆菌蛋白酶/Kex2p样前蛋白转化酶抑制剂