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- A1185 BMS-754807Target: Insulin and Insulin-like ReceptorsSummary: 有效的、选择性的IGF-1R和InsR抑制剂
- A8440 GSK1838705ATarget: Insulin and Insulin-like Receptors|ALKSummary: ATP竞争性IGF-IR/IR/ALK抑制剂
- A3608 MK 0893Target: Insulin and Insulin-like Receptors|Glucagon ReceptorsSummary: 胰高血糖素受体/ IGF-1R拮抗剂
- A3536 L-165041Target: PPARSummary: PPARβ/δ选择性激动剂
- B7797 GW 64712 CitationTarget: PPARSummary: PPARα拮抗剂
- A8601 Tankyrase Inhibitors (TNKS) 49Target: TankyrasesSummary: 端锚聚合酶抑制剂
- A2198 Genistein中文名: 金雀异黄酮,染料木素Target: Estrogen and Related Receptors|PPAR|PTKSummary: ER agonist
- B1577 C6461 CitationTarget: p300Summary: HAT p300-CBP抑制剂
- A3453 GW1929Target: PPARSummary: PPARγ激动剂
- A4305 WY-14643 (Pirinixic Acid)1 Citation中文名: 匹立尼酸Target: PPARSummary: 高效的PPARα选择性激动剂