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- A8366 ARRY-380Target: HER2Summary: 酪氨酸激酶HER2和P95-HER2抑制剂。
- B6801 SCH 79797 dihydrochlorideTarget: PARsSummary: PAR1受体拮抗剂
- A4424 SID 26681509Target: CathepsinsSummary: 人组织蛋白酶L抑制剂
- A8174 Cathepsin G Inhibitor ITarget: CathepsinsSummary: Cathepsin G抑制剂
- A1926 CA 0742 CitationTarget: CathepsinsSummary: Cathepsin B抑制剂
- A8239 CA-074 Me7 CitationTarget: CathepsinsSummary: Cathepsin B抑制剂
- A2571 Pepstatin A1 Citation中文名: 抑肽素Target: Cathepsins|Renin|HIV proteases|PepsinsSummary: 天冬氨酸蛋白酶抑制剂
- A3284 Cathepsin S inhibitor1 CitationTarget: CathepsinsSummary: 抑制MHCII抗原呈递
- A2570 Leupeptin, Microbial中文名: 亮抑酶肽Target: Cathepsins|Calpains|TrypsinsSummary: 丝氨酸和半胱氨酸蛋白酶抑制剂
- A3899 UK-50991 CitationTarget: Monocarboxylate transporters (MCTs)|mitochondrial pyruvate carrier (MPC)Summary: MCTs和MPC抑制剂