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- A3237 Betulinic acid中文名: 白桦脂酸,桦木酸Target: Aminopeptidases|Topoisomerases|HIVSummary: 抗HIV和抗肿瘤化合物,五环三萜类化合物
- A3335 Curcumin1 Citation中文名: 姜黄素Target: Histone Deacetylases (HDACs)|Nrf2|Histone Acetyltransferases (HATs)|TyrosinasesSummary: Tyrosinase(酪氨酸酶)抑制剂
- A8340 Cyclopamine1 Citation中文名: 环巴胺Target: SmoothenedSummary: Hedgehog (Hh)信号抑制剂
- B4745 (S)-10-Hydroxycamptothecin中文名: 羟喜树碱Target: TopoisomerasesSummary: 拓扑异构酶I抑制剂
- A4382 A922500Target: DGATSummary: DGAT-1抑制剂
- B2266 LDE225 (NVP-LDE225,Erismodegib)1 Citation中文名: 索尼德吉Target: SmoothenedSummary: Smoothened抑制剂
- A3215 AZD7687Target: DGATSummary: 强效的选择性DGAT抑制剂
- B3576 Omaveloxolone (RTA-408)Target: Nrf2Summary: Nrf2激活剂
- B3283 PF-04449913中文名: 格拉吉布Target: SmoothenedSummary: Smoothened拮抗剂
- A3543 LDE225 DiphosphateTarget: SmoothenedSummary: Smo拮抗剂