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- A8322 Neratinib (HKI-272)1 Citation中文名: 来那替尼Target: EGFRSummary: HER2/EGFR抑制剂
- A8555 Vandetanib (ZD6474)中文名: 凡德他尼Target: VEGFR|EGFRSummary: VEGFR2/EGFR拮抗剂
- A8199 PD153035 hydrochloride1 CitationTarget: EGFRSummary: 有效的EGFR抑制剂
- A8357 AG-1478中文名: 酪氨酸磷酸化抑制剂 AG-1478Target: EGFRSummary: EGFR抑制剂
- A3227 BAY 61-3606Target: SykSummary: Syk抑制剂
- A3823 SJB2-043Target: USPSummary: USP1抑制剂
- B2284 Fostamatinib (R788)中文名: 福坦替尼Target: SykSummary: 脾酪氨酸激酶(Syk)抑制剂
- B8023 Cerdulatinib (PRT062070)Target: JAK|Syk|TYK2Summary: Syk/JAK抑制剂
- A3736 PRT062607 Hydrochloride1 CitationTarget: SykSummary: SYK抑制剂
- B2114 Mitoxantrone HCl中文名: 米托蒽醌Target: Pim|Topoisomerases|USP|HIV IntegrasesSummary: 拓扑异构酶II抑制剂