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- A8236 Regorafenib4 Citation中文名: 瑞戈非尼Target: Raf|VEGFR|PDGFR|c-Kit|RETSummary: VEGFR/PDGFR/FGFR/mutant Kit/RET/Raf-1抑制剂
- A3750 Regorafenib hydrochloride中文名: 瑞戈非尼盐酸盐Target: Raf|VEGFR|PDGFR|c-Kit|c-RETSummary: 酪氨酸激酶抑制剂
- B5835 AZD2932Target: FLT3|VEGFR|PDGFR|c-KitSummary: VEGFR-2\PDGFRβ\Flt-3和c-Kit的抑制剂
- A8550 Telatinib (BAY 57-9352)中文名: 替拉替尼Target: VEGFR|PDGFR|c-KitSummary: VEGFR-2/-3、PDGFR-β和c-Kit抑制剂
- A2168 Dovitinib (TKI-258, CHIR-258)2 Citation中文名: 多韦替尼Target: FLT3|VEGFR|PDGFR|c-Kit|FGFRSummary: 多靶点RTK抑制剂
- A5161 Imiquimod中文名: 咪喹莫特Target: Toll-like receptors (TLRs)Summary: TLR-7激动剂,具有抗病毒和抗肿瘤活性的免疫调节剂
- A8370 Axitinib (AG 013736)1 Citation中文名: 阿西替尼Target: VEGFR|PDGFR|c-KitSummary: VEGFR1/ c-Kit抑制剂
- B5996 Motolimod (VTX-2337)Target: Toll-like receptors (TLRs)Summary: TLR8激动剂
- B5551 Poly(I:C)Target: Toll-like receptors (TLRs)Summary: Toll样受体3(TLR3)激动剂
- A3444 GS-9620中文名: 维沙莫德Target: Toll-like receptors (TLRs)Summary: TLR-7激动剂