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- A2602 Calpain Inhibitor I, ALLN2 CitationTarget: Cathepsins|CalpainsSummary: Calpain I/II/ B/L抑制剂
- A4094 MC15683 CitationTarget: Histone Deacetylases (HDACs)Summary: II类HDAC抑制剂
- A3887 Trametinib DMSO solvate1 CitationTarget: MEKSummary: 变构MEK1/MEK2 激酶抑制剂
- A4388 XL-8881 CitationTarget: HSP90Summary: Hsp90抑制剂
- A1912 Lomeguatrib中文名: 罗米鲁曲Target: O6-methylguanine-DNA-methyl-transferase (MGMT)Summary: MGMT抑制剂
- A4386 Elesclomol (STA-4783)3 Citation中文名: 伊利司莫Summary: 氧化应激/细胞凋亡诱导剂
- A2604 Celastrol中文名: 雷公藤红素Target: ProteasomeSummary: 抗氧化、抗炎和免疫抑制剂
- B1963 Lomustine1 Citation中文名: 洛莫司汀Target: RNA synthesisSummary: 抗肿瘤药
- A3723 Phloretin中文名: 根皮素Target: SGLTSummary: 在苹果中发现的二氢查耳酮
- N2771 Cepharanthine1 Citation中文名: 千金藤素Summary: 具有抗氧化活性