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- A2602 Calpain Inhibitor I, ALLN2 CitationTarget: Cathepsins|CalpainsSummary: Calpain I/II/ B/L抑制剂
- B3694 K-Ras(G12C) inhibitor 6Target: KRAS G12CSummary: K-Ras (G12C)抑制剂
- A3446 GSK1265 CitationTarget: EZH2Summary: EZH2抑制剂
- A3165 ALW-II-41-271 CitationTarget: Eph ReceptorsSummary: Eph受体抑制剂
- A8171 Entinostat (MS-275,SNDX-275)2 Citation中文名: 恩替诺特Target: Histone Deacetylases (HDACs)Summary: HDAC1和HDAC3抑制剂
- A3729 PJ34Target: PARPSummary: PARP-1抑制剂
- A8215 PP 1Target: Src|EGFR|JAK|ZAP-70Summary: Src家族酪氨酸激酶抑制剂
- A1971 Etoposide4 Citation中文名: 依托泊苷Target: TopoisomerasesSummary: 拓扑异构酶II(Topo II)抑制剂
- B5298 ABT 702 dihydrochlorideTarget: Adenosine KinasesSummary: 腺苷激酶抑制剂
- B1587 IMD 03541 CitationSummary: IKKβ抑制剂