搜索结果: 'mutant-idh1-inhibitor'
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- A3541 LCL1611 CitationTarget: Inhibitor of apoptosis proteins (IAP)Summary: IAPs拮抗剂
- A1821 Ki8751Target: VEGFRSummary: VEGFR-2有效的、选择性抑制剂
- A8641 LEE011中文名: 瑞博西利,瑞博西林Target: Cyclin-Dependent KinasesSummary: CDK4/6抑制剂
- A3209 AXL1717中文名: 鬼臼毒素Target: Insulin-like growth factor receptors(IGFRs)Summary: IGF-1R抑制剂,口服有效。
- A4383 Tolcapone中文名: 托卡朋Target: Catechol O-Methyltransferase (COMT)Summary: COMT抑制剂
- A1877 XAV-9391 CitationTarget: TNKSSummary: Tankyrase 1/2抑制剂
- B1013 GSK1324726ATarget: BromodomainsSummary: BET蛋白抑制剂
- A5112 XL147Target: PI3KSummary: PI3K选择性、可逆的抑制剂
- A8173 Romidepsin (FK228, depsipeptide)7 Citation中文名: 罗米地辛Target: Histone Deacetylases (HDACs)Summary: 选择性的HDAC1/HDAC2抑制剂