搜索结果: 'inhibitors-and-substrate'
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- A3149 AKT inhibitor VIII2 CitationTarget: AktSummary: 变构Akt激酶抑制剂
- A8623 TOK-001中文名: 加来特龙,伽来特隆Target: Androgen Receptors|Cytochrome P450 (CYP450)Summary: CYP17抑制剂和雄激素受体(AR)拮抗剂
- A3003 MDV3100 (Enzalutamide)12 Citation中文名: 恩杂鲁胺Target: Androgen ReceptorsSummary: 雄激素受体拮抗剂。
- A2150 AndarineTarget: Androgen ReceptorsSummary: 雄激素受体拮抗剂
- A5065 Bicalutamide1 Citation中文名: 比卡鲁胺Target: Androgen ReceptorsSummary: 雄激素受体(Androgen receptor)拮抗剂
- B2180 AS-252424Target: Akt|PI3KSummary: PI3Kγ抑制剂
- A5653 AT7867Target: Akt|PKA|p70 rskSummary: Akt1/2/3和p70S6K/PKA的抑制剂
- A5072 GSK690693Target: Akt|PKC|PKG|PKA|PrkSummary: ATP竞争性的Pan-AKT抑制剂
- A8499 PF-04691502Target: Akt|PI3K|mTORSummary: PI3K/mTOR (FRAP)抑制剂
- A3006 GDC-0068 (RG7440)Target: AktSummary: Pan-AKT抑制剂