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- A1905 3-Deazaneplanocin,DZNep6 Citation中文名: 3-去氮腺嘌呤ATarget: HydrolaseSummary: S-腺苷高半胱氨酸和EZH2抑制剂。
- A8182 3-Deazaneplanocin A (DZNep) hydrochloride1 Citation中文名: 3-去氮腺嘌呤A盐酸盐Target: EZH2Summary: SAHH和EZH2抑制剂
- A3011 CHIR-99021 (CT99021)2 CitationTarget: GSK-3Summary: GSK-3抑制剂
- A8350 AZD4547Target: FGFRSummary: FGFR抑制剂
- B6020 GSK6211 CitationTarget: AMPKSummary: AMPK激动剂
- B2266 LDE225 (NVP-LDE225,Erismodegib)1 Citation中文名: 索尼德吉Target: SmoothenedSummary: Smoothened抑制剂
- B2193 Mitiglinide Calcium中文名: 米格列奈钙Target: Inward Rectifier Potassium (Kir) ChannelsSummary: 钾通道抑制剂
- A3843 SU 5402Target: VEGFR|PDGFR|FGFRSummary: VEGFR2/FGFR/PDGFR/EGFR抑制剂
- A5801 BIX 02189Target: MEK|ERKSummary: MEK5抑制剂
- A8335 Palbociclib (PD0332991) Isethionate1 Citation中文名: 帕博西尼羟乙基磺酸盐Target: Cyclin-Dependent KinasesSummary: CDK4/6抑制剂