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- B7070 Triacsin CTarget: Synthases/SynthetasesSummary: 酰基辅酶A合成酶抑制剂
- A4127 GSK1070916Target: Aurora KinasesSummary: Aurora B/C抑制剂
- A3020 (R)-Crizotinib2 Citation中文名: 克唑替尼Target: c-METSummary: ATP竞争性的C-MET/ALK抑制剂。
- A3183 Ansamitocin P-3中文名: 安丝菌素 P 3'Target: Microtubules/TubulinsSummary: 美登素类似物,微管蛋白抑制剂
- A5703 BMS-777607Target: METSummary: 强效的c-Met选择性抑制剂
- A3632 Motesanib中文名: 莫特塞尼Target: VEGFRSummary: Flk-1/Flt-4/PDGFR-/c-Kit抑制剂
- N2791 Cucurbitacin E中文名: 葫芦素 ETarget: ActinSummary: 抑制肌动蛋白解聚
- N1375 Solamargine中文名: 澳洲茄边碱,边缘茄碱Summary: 细胞毒性剂
- B7207 SecinH3Target: Guanine nucleotide exchange factors (GEFs)Summary: Sec7特异性GEF抑制剂
- N2771 Cepharanthine1 Citation中文名: 千金藤素Summary: 具有抗氧化活性