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- A3927 VS-5584 (SB2343)Target: PI3K|mTORSummary: MTOR/P13K抑制剂
- A4390 Pemetrexed1 Citation中文名: 培美曲塞二钠盐Target: Thymidylate Synthase|DHFR|GARFTSummary: TS、DHFR、GARFT和AICARFT抑制剂
- A8808 ME0328Target: PARPSummary: PARP抑制剂
- A3729 PJ34Target: PARPSummary: PARP-1抑制剂
- A4160 A-966492Target: PARPSummary: PARP-1/-2抑制剂
- A3617 MK-4827中文名: 尼拉帕尼Target: PARPSummary: PARP-1/-2抑制剂
- A5112 XL147Target: PI3KSummary: PI3K选择性、可逆的抑制剂
- A8554 Dapivirine (TMC120)中文名: 达匹维林Target: Reverse TranscriptasesSummary: 非核苷逆转录酶抑制剂
- A4163 UPF 1069Target: PARPSummary: PARP2选择性抑制剂
- A3958 Veliparib dihydrochloride中文名: 维利帕尼二盐酸盐Target: PARPSummary: PARP-1/PARP-2抑制剂