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- A2942 Masitinib (AB1010)中文名: 马赛替尼Target: PDGFR|c-Kit|LynSummary: 酪氨酸激酶抑制剂
- B2219 EHop-0161 CitationTarget: RacSummary: Rac1/Rac3 GTPase抑制剂
- A2249 T0901317Target: Liver X receptors (LXRs)Summary: 肝X受体激动剂
- A8808 ME0328Target: PARPSummary: PARP抑制剂
- A3729 PJ34Target: PARPSummary: PARP-1抑制剂
- A4160 A-966492Target: PARPSummary: PARP-1/-2抑制剂
- A3617 MK-4827中文名: 尼拉帕尼Target: PARPSummary: PARP-1/-2抑制剂
- A4163 UPF 1069Target: PARPSummary: PARP2选择性抑制剂
- A3958 Veliparib dihydrochloride中文名: 维利帕尼二盐酸盐Target: PARPSummary: PARP-1/PARP-2抑制剂
- A8394 CHIR-124Target: FLT3|GSK-3|Chk|PDGFRSummary: Chk1抑制剂