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- A8177 PAC-11 CitationTarget: CaspasesSummary: 半胱天冬酶-3酶原激活剂
- A8803 RGFP9664 CitationTarget: Histone Deacetylases (HDACs)Summary: HDAC3抑制剂
- A3573 LY2801653Target: METSummary: MET抑制剂
- A8393 CH5424802中文名: 阿来替尼Target: ALKSummary: ALK的有效ATP竞争性抑制剂
- A4210 Bay 11-7821(BAY 11-7082)1 CitationSummary: IKK/NF-κB/TNFα抑制剂
- A4381 FK866 (APO866)1 Citation中文名: 达珀利奈Target: NamptSummary: NAMPT抑制剂
- B3697 4E1RCatTarget: eIF4FSummary: eIF4E:eIF4G与eIF4E:4E-BP1相互作用的双重抑制剂
- A1670 Enzastaurin (LY317615)2 Citation中文名: 恩扎妥林Target: PKCSummary: PKCβ抑制剂
- A1933 Carfilzomib (PR-171)10 Citation中文名: 卡非佐米Target: ProteasomeSummary: 蛋白酶体抑制剂
- A4171 EPZ0056872 CitationTarget: EZH2Summary: EZH2抑制剂