P-gp
P-gp (P-glycoprotein) is a ATP-binding cassette transproters which overepxressed in multidrug-resistance cancer cells. It functions in pumping drug out of cell and lower intracellular drug concentration.
- C3840 Estradiol 17-(β-D-Glucuronide) (sodium salt)Summary: 多药耐药蛋白2(MRP2)的底物
- C3897 Estradiol 3-(β-D-Glucuronide) (sodium salt)Summary: 多药耐药蛋白2(MRP2)的底物
- C3610 HypophyllanthinSummary: P-糖蛋白(P-gp)抑制剂
- C3140 Rhodamine 123 (chloride)Summary: 膜可渗透的阳离子染料,用作流出泵P-糖蛋白的底物
- B1167 Dofequidar fumarateSummary: MDR逆转剂
- A8549 LY335979 (Zosuquidar 3HCL)1 CitationTarget: P-glycoprotein (P-gp)Summary: Pgb(P糖蛋白)抑制剂
- A3956 ZosuquidarTarget: P-glycoprotein (P-gp)|Cytochrome P450 (CYP450)Summary: MDR调节剂
- A3859 Tariquidar methanesulfonate, hydrateTarget: P-glycoprotein (P-gp)Summary: P-糖蛋白抑制剂
- A8208 Tariquidar2 CitationTarget: P-glycoprotein (P-gp)Summary: P-糖蛋白抑制剂