Cyclin-Dependent Kinases
Cyclin-dependent kinases is a group of serine/threonine kinases. It is activated by binding to cyclin and participates in the regulation of cell cycle.
- B7855 AlsterpaulloneSummary: CDKs和GSK3β抑制剂
- C4040 OlomoucineSummary: cdk抑制剂
- C3767 Iso-OlomoucineSummary: Cdk5抑制剂奥洛莫辛(olomoucine)的无活性立体异构体
- C3679 Cdk1/2 Inhibitor IIISummary: Cdk1/细胞周期蛋白B和Cdk2/细胞周期蛋白A抑制剂
- C3995 Cdk4/6 Inhibitor IVSummary: Cdk4/cyclin D1和Cdk6/cyclin D1抑制剂
- B6192 ON123300Summary: 多靶点激酶抑制剂,抑制CDK4,Ark5,PDGFRβ,FGFR1,RET和Fyn。
- B6101 BohemineSummary: CDK抑制剂
- A8739 CCT251545 analogue, Compound 51Summary: CDK8/CDK19的强效选择性抑制剂,具有口服活性
- A8736 THZ531Target: Cyclin-Dependent KinasesSummary: CDK12 和CDK13共价抑制剂
- A8732 Senexin BSummary: CDK8/CDK19的强效选择性抑制剂,具有口服活性