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Signaling Pathways - DNA Alkylating - Smoothened - sodium channel

10 件产品

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  1. Ibutilide Fumarate
    B2278 Ibutilide Fumarate
    中文名: 富马酸伊布利特
    Target: Voltage-gated Potassium (KV) Channels|Voltage-gated Calcium Channels (CaV)|sodium channel
    Summary: III类抗心律失常药物
      ≥25.6 mg/mL
      ≥16.4 mg/mL
  2. Lamotrigine
    B2249 Lamotrigine
     1 Citation
    中文名: 拉莫三嗪
    Target: 5-HT receptors|sodium channel
    Summary: 5-HT抑制剂,钠通道阻断剂
      ≥12.3 mg/mL
      insoluble in H2O
  3. LDE225 (NVP-LDE225,Erismodegib)
    B2266 LDE225 (NVP-LDE225,Erismodegib)
     1 Citation
    中文名: 索尼德吉
    Target: Smoothened
    Summary: Smoothened抑制剂
      ≥24.3 mg/mL
      insoluble in H2O
  4. PF-04449913
    B3283 PF-04449913
    中文名: 格拉吉布
    Target: Smoothened
    Summary: Smoothened拮抗剂
      ≥20.15 mg/mL
      insoluble in H2O
  5. Cyclopamine
    A8340 Cyclopamine
     1 Citation
    中文名: 环巴胺
    Target: Smoothened
    Summary: Hedgehog (Hh)信号抑制剂
      ≥6.86 mg/mL
      insoluble in H2O
  6. Ifosfamide
    A2097 Ifosfamide
    中文名: 异环磷酰胺
    Target: DNA Alkylating
    Summary: 细胞抑制剂
      ≥13.05 mg/mL
      ≥22 mg/mL
  7. Dacarbazine
    A2197 Dacarbazine
    中文名: 达卡巴嗪
    Target: DNA Alkylating
    Summary: 抗肿瘤(恶性黑色素瘤和肉瘤)
      ≥2.28 mg/mL
      ≥0.54 mg/mL
  8. LDE225 Diphosphate
    A3543 LDE225 Diphosphate
    Target: Smoothened
    Summary: Smo拮抗剂
      ≥27.85 mg/mL
      insoluble in H2O
  9. Dronedarone
    A3374 Dronedarone
    中文名: 决奈达隆
    Target: Cytochrome P450 (CYP450)|sodium channel|adrenergic receptor|potassium channel|calcium channel
    Summary: CYP3A4和2D6抑制剂
      ≥27.84 mg/mL
      insoluble in H2O
  10. BMS-833923
    A3258 BMS-833923
    Target: Smoothened
    Summary: Smoothened抑制剂
      ≥47.4 mg/mL
      insoluble in H2O

10 件产品

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