Signaling Pathways - Calcium-Sensing Receptors (CaSRs) - Ub-conjugating enzyme (E2) complex - G9a - p53
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- B7757 UNC 0642Target: G9a|GLPSummary: G9a和GLP组蛋白赖氨酸甲基转移酶抑制剂
- B7504 R 568 hydrochlorideTarget: Calcium-Sensing Receptors (CaSRs)Summary: 人类钙敏感受体(hCaSR)的正变构调节剂
- A8813 NSC697923Target: Ub-conjugating enzyme (E2) complexSummary: E2复合体Ubc13-Uev1A抑制剂
- A4482 Pifithrin-μ1 CitationTarget: Autophagy|p53|HSP70Summary: p53结合抑制剂,抗凋亡。
- A4483 PRIMA-1Target: p53Summary: BAX抑制剂
- A4481 PhiKan 083Target: p53Summary: P53稳定剂
- A3667 NPS-2143 hydrochlorideTarget: Calcium-Sensing Receptors (CaSRs)Summary: 钙离子敏感受体拮抗剂
- A1909 BIX 01294Target: G9aSummary: G9a和GLP抑制剂
- A4203 Tenovin-1Target: Sir2-like Family Deacetylases (Sirtuins)|p53|p21Summary: SIRT2 抑制剂,p53激活剂
- A4204 JNJ-26854165 (Serdemetan)1 CitationTarget: p53|HDM2 ubiquitin ligaseSummary: P53激活剂,阻断Mdm2-p53相互作用。