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Signaling Pathways - sodium channel - Serotonin reuptake - SETD7 - Tie-2

10 件产品

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  1. Pexmetinib (ARRY-614)
    B6012 Pexmetinib (ARRY-614)
    Target: p38|Tie-2
    Summary: p38 MAPK 和 Tie2/Tek 受体酪氨酸激酶的双重抑制剂
      ≥107.6 mg/mL
      insoluble in H2O
  2. Altiratinib
    B5832 Altiratinib
     1 Citation
    Target: FLT3|VEGFR|Trk Receptors|c-MET|Tie-2
    Summary: c-MET/TIE-2/VEGFR抑制剂
      ≥21.55 mg/mL
      insoluble in H2O
  3. ACTB-1003
    B4904 ACTB-1003
    Target: VEGFR|FGFR|Tie-2|RSK|p70 S6K
    Summary: FGFR1抑制剂
      ≥18.15 mg/mL
      insoluble in H2O
  4. PFI-2
    B4875 PFI-2
     1 Citation
    Target: SETD7
    Summary: SETD7甲基转移酶抑制剂
      ≥50 mg/mL
      ≥1.51 mg/mL
  5. Ibutilide Fumarate
    B2278 Ibutilide Fumarate
    中文名: 富马酸伊布利特
    Target: Voltage-gated Potassium (KV) Channels|Voltage-gated Calcium Channels (CaV)|sodium channel
    Summary: III类抗心律失常药物
      ≥25.6 mg/mL
      ≥16.4 mg/mL
  6. Lamotrigine
    B2249 Lamotrigine
     1 Citation
    中文名: 拉莫三嗪
    Target: 5-HT receptors|sodium channel
    Summary: 5-HT抑制剂,钠通道阻断剂
      ≥12.3 mg/mL
      insoluble in H2O
  7. Fluvoxamine
    B1205 Fluvoxamine
    中文名: 氟伏沙明
    Target: Serotonin reuptake
    Summary: 选择性5-羟色胺再摄取抑制剂
      ≥15.92 mg/mL
      insoluble in H2O
  8. DCC-2036 (Rebastinib)
    B1404 DCC-2036 (Rebastinib)
    Target: FLT3|Bcr-Abl|Tie-2|KDR
    Summary: Bcr-Abl抑制剂
      ≥27.7 mg/mL
  9. Tie2 kinase inhibitor
    A5979 Tie2 kinase inhibitor
    中文名: Tie2激酶抑制剂
    Target: Tie-2
    Summary: Tie-2(Tie2 )抑制剂
      ≥22 mg/mL
      insoluble in H2O
  10. Dronedarone
    A3374 Dronedarone
    中文名: 决奈达隆
    Target: Cytochrome P450 (CYP450)|sodium channel|adrenergic receptor|potassium channel|calcium channel
    Summary: CYP3A4和2D6抑制剂
      ≥27.84 mg/mL
      insoluble in H2O

10 件产品

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