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Signaling Pathways - SMARCA2 - GSK-3 - Cytochrome P450 (CYP450)

26件产品中的 1-10

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  1. 7-Ethoxyresorufin
    B5963 7-Ethoxyresorufin
    中文名: 乙氧基试卤灵,7-乙氧基-3H-吩恶嗪-3-酮
    Target: Cytochrome P450 (CYP450)
    Summary: CYP1A特异性底物
      Soluble in DMSO
  2. Bikinin
    B4898 Bikinin
    Target: GSK-3
    Summary: GSK3抑制剂和油菜素类固醇激活剂
      ≥13.65 mg/mL
      insoluble in H2O
  3. PFI 3
    B7744 PFI 3
    Target: Protein polybromo-1|SMARCA4|SMARCA2
    Summary: Polybromo 1和SMARCA4抑制剂
      ≥15.15 mg/mL
      insoluble in H2O
  4. Quinidine
    B7590 Quinidine
    中文名: 奎尼丁
    Target: Voltage-gated Sodium (NaV) Channels|Cytochrome P450 (CYP450)
    Summary: 降低Na+和K+通道电流
      ≥11.95 mg/mL
      insoluble in H2O
  5. Indirubin
    B3672 Indirubin
    中文名: 靛玉红
    Target: Cyclin-Dependent Kinases|GSK-3
    Summary: 细胞周期蛋白依赖性激酶和GSK-3β抑制剂
      ≥13.1 mg/mL
      insoluble in H2O
  6. Fluconazole
    B2094 Fluconazole
    中文名: 氟康唑
    Target: Cytochrome P450 (CYP450)
    Summary: 三唑抗真菌剂
      ≥10.9 mg/mL
      insoluble in H2O
  7. Rifabutin
    B2126 Rifabutin
    中文名: 利福布丁
    Target: Cytochrome P450 (CYP450)
    Summary: 抗结核药物
      ≥42.35 mg/mL
      insoluble in H2O
  8. AZD1080
    B1536 AZD1080
     1 Citation
    Target: GSK-3
    Summary: GSK3β抑制剂
      ≥16.7 mg/mL
      insoluble in H2O
  9. TOK-001
    A8623 TOK-001
    中文名: 加来特龙,伽来特隆
    Target: Androgen Receptors|Cytochrome P450 (CYP450)
    Summary: CYP17抑制剂和雄激素受体(AR)拮抗剂
      ≥12.4 mg/mL
      insoluble in H2O
  10. A-674563
    A8616 A-674563
    Target: Cyclin-Dependent Kinases|Akt|GSK-3|ERK|PKC|PKA|RSK
    Summary: Akt1 / PKA / CDK2的强效选择性抑制剂
      ≥4.9 mg/mL
      ≥23.8 mg/mL

26件产品中的 1-10

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