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Signaling Pathways - endothelin receptor - M3 Receptors - 5-HT7 Receptors - PKA

16件产品中的 1-10

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  1. FR 139317
    B5082 FR 139317
    Target: endothelin receptor
    Summary: 选择性ETA内皮素受体拮抗剂
      Soluble to 100 mM in 1eq. HCl and to 100 mM in DMSO
  2. H-7 dihydrochloride
    B6342 H-7 dihydrochloride
    Target: PKC|PKG|PKA|Myosin light chain kinases (MLCKs)
    Summary: 蛋白激酶抑制剂
      Soluble in DMSO
  3. Midostaurin (PKC412)
    B3709 Midostaurin (PKC412)
    中文名: 米哚妥林
    Target: PKC|PKA|KDR|Flk1|PPK|c-Syk|CDK1/CyclinB
    Summary: PKC抑制剂
      ≥57.1 mg/mL
      insoluble in H2O
  4. 8-Bromo-cAMP, sodium salt
    B9000 8-Bromo-cAMP, sodium salt
    中文名: 8-溴腺苷3',5'-环腺苷一磷酸
    Target: PKA
    Summary: 细胞渗透性cAMP类似物,激活PKA
      ≥22.43 mg/mL
      ≥43 mg/mL
  5. Fasudil
    B3523 Fasudil
    中文名: 法舒地尔
    Target: ROCK|PKC|PKG|PKA|Myosin light chain kinases (MLCKs)
    Summary: 钙拮抗剂
      Soluble in DMSO
  6. Otilonium Bromide
    B1607 Otilonium Bromide
    中文名: 奥替溴铵
    Target: M3 Receptors
    Summary: AChR抑制剂
      ≥28.18 mg/mL
      ≥55.8 mg/mL
  7. Lurasidone HCl
    B1477 Lurasidone HCl
    中文名: 盐酸鲁拉西酮
    Target: 5-HT2 Receptors|D2 Receptors|5-HT1 Receptors|5-HT7 Receptors
    Summary: 多巴胺D2/5-HT2A/5-HT7/5-HT1A抑制剂
      ≥11.11 mg/mL
      insoluble in H2O
  8. Quetiapine Fumarate
    B1490 Quetiapine Fumarate
     1 Citation
    中文名: 富马酸奎硫平
    Target: 5-HT2 Receptors|D1 and D5 Receptors|D2 Receptors|D3 Receptors|5-HT1 Receptors|5-HT7 Receptors
    Summary: 多巴胺受体拮抗剂
      ≥11.03 mg/mL
      insoluble in H2O
  9. Darifenacin HBr
    B1600 Darifenacin HBr
    中文名: 氢溴酸达非那新
    Target: M3 Receptors
    Summary: 选择性M3毒蕈碱受体拮抗剂
      ≥20.2 mg/mL
      insoluble in H2O
  10. Solifenacin succinate
    B1614 Solifenacin succinate
    中文名: 琥珀酸索非那新
    Target: M3 Receptors
    Summary: 毒蕈碱受体拮抗剂
      ≥24.05 mg/mL
      ≥53.6 mg/mL

16件产品中的 1-10

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