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Signaling Pathways - Nuclear Receptors - Farnesoid X receptors (FXRs) - PKG - Estrogen and Related Receptors

18件产品中的 1-10

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  1. Obeticholic Acid
    B4888 Obeticholic Acid
     2 Citation
    中文名: 奥贝胆酸
    Target: Farnesoid X receptors (FXRs)
    Summary: FXR激动剂
      ≥21.5 mg/mL
      insoluble in H2O
  2. (Z)-4-Hydroxytamoxifen
    B5421 (Z)-4-Hydroxytamoxifen
    中文名: 4-羟基他莫昔芬
    Target: Estrogen and Related Receptors
    Summary: 雌激素受体(ER)调节剂
      ≥38.8 mg/mL
      insoluble in H2O
  3. H-7 dihydrochloride
    B6342 H-7 dihydrochloride
    Target: PKC|PKG|PKA|Myosin light chain kinases (MLCKs)
    Summary: 蛋白激酶抑制剂
      Soluble in DMSO
  4. DLPC
    B7661 DLPC
    Target: Nuclear Receptors
    Summary: LRH-1激动剂配体
      insoluble in DMSO
      insoluble in H2O
  5. Fasudil
    B3523 Fasudil
    中文名: 法舒地尔
    Target: ROCK|PKC|PKG|PKA|Myosin light chain kinases (MLCKs)
    Summary: 钙拮抗剂
      Soluble in DMSO
  6. Erteberel (LY500307)
    B1518 Erteberel (LY500307)
    Target: Estrogen and Related Receptors
    Summary: ERβ激动剂
      ≥14.1 mg/mL
      insoluble in H2O
  7. Estriol
    B1507 Estriol
    中文名: 雌三醇
    Target: Estrogen and Related Receptors
    Summary: 雌激素受体拮抗剂
      ≥9.25 mg/mL
      insoluble in H2O
  8. Estradiol valerate
    B1506 Estradiol valerate
    中文名: 戊酸雌二醇
    Target: Estrogen and Related Receptors
    Summary: 雌激素受体激动剂
      ≥15.45 mg/mL
      insoluble in H2O
  9. Bazedoxifene HCl
    B1519 Bazedoxifene HCl
    中文名: 盐酸巴多昔芬
    Target: Estrogen and Related Receptors
    Summary: 新的非甾体,基于吲哚的雌激素受体调节剂(SERM)
      ≥25.35 mg/mL
  10. Toremifene Citrate
    B1513 Toremifene Citrate
    中文名: 枸橼酸托瑞米芬
    Target: Estrogen and Related Receptors
    Summary: 口服选择性雌激素受体调节剂(SERM)
      ≥24.15 mg/mL
      insoluble in H2O

18件产品中的 1-10

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