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Signaling Pathways - cAMP - Squalene epoxidases - Delayed rectifier outward potassium current (IKr) - NAE - Cytochrome P450 (CYP450)

22件产品中的 1-10

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  1. 7-Ethoxyresorufin
    B5963 7-Ethoxyresorufin
    中文名: 乙氧基试卤灵,7-乙氧基-3H-吩恶嗪-3-酮
    Target: Cytochrome P450 (CYP450)
    Summary: CYP1A特异性底物
      Soluble in DMSO
  2. Quinidine
    B7590 Quinidine
    中文名: 奎尼丁
    Target: Voltage-gated Sodium (NaV) Channels|Cytochrome P450 (CYP450)
    Summary: 降低Na+和K+通道电流
      ≥11.95 mg/mL
      insoluble in H2O
  3. Tolbutamide
    B2194 Tolbutamide
    中文名: 甲苯磺丁脲
    Target: cAMP|Sulfonylurea receptors
    Summary: 第一代钾通道阻滞剂
      ≥10.05 mg/mL
      insoluble in H2O
  4. Fluconazole
    B2094 Fluconazole
    中文名: 氟康唑
    Target: Cytochrome P450 (CYP450)
    Summary: 三唑抗真菌剂
      ≥10.9 mg/mL
      insoluble in H2O
  5. MLN4924
    B1036 MLN4924
     5 Citation
    Target: NAE|Ubiquitin-activating Enzyme E1|SUMOylation
    Summary: NAE抑制剂
      ≥22.18 mg/mL
      insoluble in H2O
  6. Butenafine HCl
    B1901 Butenafine HCl
    中文名: 盐酸布替萘芬
    Target: Squalene epoxidases
    Summary: 合成苄胺抗真菌剂
      ≥17.55 mg/mL
      insoluble in H2O
  7. Terbinafine HCl
    B2047 Terbinafine HCl
    中文名: 盐酸特比萘芬
    Target: Squalene epoxidases
    Summary: 有效的非竞争性角鲨烯环氧酶抑制剂
      ≥16.3 mg/mL
      insoluble in H2O
  8. Rifabutin
    B2126 Rifabutin
    中文名: 利福布丁
    Target: Cytochrome P450 (CYP450)
    Summary: 抗结核药物
      ≥42.35 mg/mL
      insoluble in H2O
  9. TOK-001
    A8623 TOK-001
    中文名: 加来特龙,伽来特隆
    Target: Androgen Receptors|Cytochrome P450 (CYP450)
    Summary: CYP17抑制剂和雄激素受体(AR)拮抗剂
      ≥12.4 mg/mL
      insoluble in H2O
  10. Dofetilide
    A8417 Dofetilide
     2 Citation
    中文名: 多非利特
    Target: Delayed rectifier outward potassium current (IKr)
    Summary: 钾通道抑制剂
      ≥21.15 mg/mL
      insoluble in H2O

22件产品中的 1-10

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