Signaling Pathways - cAMP - Squalene epoxidases - Delayed rectifier outward potassium current (IKr) - NAE - Cytochrome P450 (CYP450)
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- B5963 7-Ethoxyresorufin中文名: 乙氧基试卤灵,7-乙氧基-3H-吩恶嗪-3-酮Target: Cytochrome P450 (CYP450)Summary: CYP1A特异性底物
- B7590 Quinidine中文名: 奎尼丁Target: Voltage-gated Sodium (NaV) Channels|Cytochrome P450 (CYP450)Summary: 降低Na+和K+通道电流
- B2194 Tolbutamide中文名: 甲苯磺丁脲Target: cAMP|Sulfonylurea receptorsSummary: 第一代钾通道阻滞剂
- B2094 Fluconazole中文名: 氟康唑Target: Cytochrome P450 (CYP450)Summary: 三唑抗真菌剂
- B1036 MLN49245 CitationTarget: NAE|Ubiquitin-activating Enzyme E1|SUMOylationSummary: NAE抑制剂
- B1901 Butenafine HCl中文名: 盐酸布替萘芬Target: Squalene epoxidasesSummary: 合成苄胺抗真菌剂
- B2047 Terbinafine HCl中文名: 盐酸特比萘芬Target: Squalene epoxidasesSummary: 有效的非竞争性角鲨烯环氧酶抑制剂
- B2126 Rifabutin中文名: 利福布丁Target: Cytochrome P450 (CYP450)Summary: 抗结核药物
- A8623 TOK-001中文名: 加来特龙,伽来特隆Target: Androgen Receptors|Cytochrome P450 (CYP450)Summary: CYP17抑制剂和雄激素受体(AR)拮抗剂
- A8417 Dofetilide2 Citation中文名: 多非利特Target: Delayed rectifier outward potassium current (IKr)Summary: 钾通道抑制剂