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Signaling Pathways - BCPCF efflux - Myosin light chain kinases (MLCKs) - O6-methylguanine-DNA-methyl-transferase (MGMT) - DNA Methyltransferases

10 件产品

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  1. Sodium Tauroursodeoxycholate (TUDC)
    B6019 Sodium Tauroursodeoxycholate (TUDC)
    中文名: 牛磺熊去氧胆酸钠
    Target: BCPCF efflux
    Summary: 水溶性胆汁盐
      ≥26.1 mg/mL
      ≥8.42 mg/mL
  2. Procainamide HCl
    B4798 Procainamide HCl
    中文名: 盐酸普鲁卡因胺
    Target: DNA Methyltransferases
    Summary: 钠通道阻滞剂
      ≥13.65 mg/mL
      ≥46.4 mg/mL
  3. H-7 dihydrochloride
    B6342 H-7 dihydrochloride
    Target: PKC|PKG|PKA|Myosin light chain kinases (MLCKs)
    Summary: 蛋白激酶抑制剂
      Soluble in DMSO
  4. Fasudil
    B3523 Fasudil
    中文名: 法舒地尔
    Target: ROCK|PKC|PKG|PKA|Myosin light chain kinases (MLCKs)
    Summary: 钙拮抗剂
      Soluble in DMSO
  5. ML-7 hydrochloride
    A3626 ML-7 hydrochloride
    Target: Myosin light chain kinases (MLCKs)
    Summary: 肌球蛋白轻链激酶抑制剂
      ≥15.95 mg/mL
      ≥8.82 mg/mL
  6. Zebularine
    A1915 Zebularine
     1 Citation
    中文名: 泽布拉林
    Target: DNA Methyltransferases|Cytidine deaminases
    Summary: DNA甲基化抑制剂
      ≥8.3 mg/mL
      ≥50.7 mg/mL
  7. RG 108
    A1913 RG 108
     3 Citation
    Target: DNA Methyltransferases
    Summary: DNA甲基转移酶抑制剂
      ≥16.7 mg/mL
      insoluble in H2O
  8. Lomeguatrib
    A1912 Lomeguatrib
    中文名: 罗米鲁曲
    Target: O6-methylguanine-DNA-methyl-transferase (MGMT)
    Summary: MGMT抑制剂
      ≥50 mg/mL
      insoluble in H2O
  9. 5-Azacytidine
    A1907 5-Azacytidine
     6 Citation
    中文名: 氮胞苷(5-氮胞苷)
    Target: DNA Methyltransferases
    Summary: DNA甲基转移酶抑制剂
      ≥24.45 mg/mL
      ≥13.55 mg/mL
  10. Parthenolide
    N1315 Parthenolide
    中文名: 小白菊内酯,欧苷菊
    Target: Histone Deacetylases (HDACs)|MDM2|DNA Methyltransferases|p53|5-HT
      ≥9.2 mg/mL
      insoluble in H2O

10 件产品

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