Signaling Pathways - ROS1 - Flk1 - G-quadruplexes - Nrf2
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- B5859 Entrectinib中文名: 恩曲替尼Target: Trk Receptors|ALK|ROS1Summary: ALK激酶抑制剂
- B4882 PF-06463922中文名: 劳拉替尼Target: ALK|ROS1Summary: ALK/ROS1的强效选择性抑制剂
- B3709 Midostaurin (PKC412)中文名: 米哚妥林Target: PKC|PKA|KDR|Flk1|PPK|c-Syk|CDK1/CyclinBSummary: PKC抑制剂
- B3576 Omaveloxolone (RTA-408)Target: Nrf2Summary: Nrf2激活剂
- A2597 Brivanib (BMS-540215)中文名: 布立尼布Target: VEGFR|FGFR|Flk1Summary: VEGFR-2的ATP竞争性抑制剂
- A3742 Pyridostatin2 CitationTarget: G-quadruplexesSummary: 促生长停滞药物
- A3335 Curcumin1 Citation中文名: 姜黄素Target: Histone Deacetylases (HDACs)|Nrf2|Histone Acetyltransferases (HATs)|TyrosinasesSummary: Tyrosinase(酪氨酸酶)抑制剂
- A3221 Bardoxolone methyl中文名: 甲基巴多索隆Target: Nrf2Summary: IKK抑制剂,强效的抗氧化炎性反应调节剂。