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Signaling Pathways - ROS1 - Notch - 5-HT receptor - Calpains

10 件产品

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  1. Entrectinib
    B5859 Entrectinib
    中文名: 恩曲替尼
    Target: Trk Receptors|ALK|ROS1
    Summary: ALK激酶抑制剂
      ≥28.05 mg/mL
      insoluble in H2O
  2. PF-06463922
    B4882 PF-06463922
    中文名: 劳拉替尼
    Target: ALK|ROS1
    Summary: ALK/ROS1的强效选择性抑制剂
      ≥20.3 mg/mL
      insoluble in H2O
  3. Latrepirdine
    B1572 Latrepirdine
    Target: Voltage-gated Calcium Channels (CaV)|NMDA receptor|adrenergic receptor|Histamine receptors|GluR|5-HT receptor|dopamine receptors|AMPA receptor
    Summary: 脑细胞死亡抑制剂
      ≥19.62 mg/mL
      insoluble in H2O
  4. PD 150606
    A4413 PD 150606
    Target: Calpains
    Summary: 非肽类钙蛋白酶抑制剂
      Soluble in DMSO
  5. MDL 28170
    A4412 MDL 28170
    Target: Cathepsins|Calpains
    Summary: Calpain和cathepsin B抑制剂
      ≥16.75 mg/mL
      insoluble in H2O
  6. Quetiapine
    A3744 Quetiapine
    中文名: 喹硫平
    Target: AChR|adrenergic receptor|5-HT receptor|Dopamine receptor|Histamine receptor
    Summary: 多巴胺受体拮抗剂
      ≥19.18 mg/mL
      insoluble in H2O
  7. LY3039478
    A4023 LY3039478
     1 Citation
    Target: Notch
    Summary: Notch抑制剂
      ≥23.2 mg/mL
      insoluble in H2O
  8. Calpain Inhibitor I, ALLN
    A2602 Calpain Inhibitor I, ALLN
     2 Citation
    Target: Cathepsins|Calpains
    Summary: Calpain I/II/ B/L抑制剂
      ≥19.1 mg/mL
      insoluble in H2O
  9. E-64
    A2576 E-64
     2 Citation
    Target: Cathepsins|Calpains|Papains
    Summary: 半胱氨酸蛋白酶(cysteine protease)抑制剂
      ≥53.6 mg/mL
      ≥49.1 mg/mL
  10. Leupeptin, Microbial
    A2570 Leupeptin, Microbial
    中文名: 亮抑酶肽
    Target: Cathepsins|Calpains|Trypsins
    Summary: 丝氨酸和半胱氨酸蛋白酶抑制剂
      ≥24.7 mg/mL
      ≥54.4 mg/mL

10 件产品

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