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Signaling Pathways - SGLT - DPP-4 - Calcium-Activated Potassium (KCa) Channels

10 件产品

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  1. Talabostat mesylate
    B3941 Talabostat mesylate
     2 Citation
    Target: DPP-4
    Summary: DPP4抑制剂
      ≥11.45 mg/mL
      ≥31 mg/mL
  2. Dequalinium Chloride
    B2191 Dequalinium Chloride
    中文名: 地喹氯铵
    Target: PKC|Calcium-Activated Potassium (KCa) Channels
    Summary: PKC抑制剂
      insoluble in DMSO
      insoluble in H2O
  3. Saxagliptin
    A8650 Saxagliptin
    中文名: 沙格列汀
    Target: DPP-4
    Summary: DPP4抑制剂
      ≥14.85 mg/mL
      ≥8.32 mg/mL
  4. Canagliflozin
    A8333 Canagliflozin
     1 Citation
    中文名: 卡格列净
    Target: SGLT
    Summary: SGLT2的有效选择性抑制剂
      ≥22.25 mg/mL
      insoluble in H2O
  5. Zonisamide
    A5354 Zonisamide
    中文名: 唑尼沙胺
    Target: Voltage-gated Sodium (NaV) Channels|Voltage-gated Calcium Channels (CaV)|Carbonic Anhydrases|Calcium-Activated Potassium (KCa) Channels
    Summary: 抗惊厥和机械效应的抗癫痫药
      ≥8.35 mg/mL
      insoluble in H2O
  6. TRAM-34
    A1888 TRAM-34
    Target: Calcium-Activated Potassium (KCa) Channels
    Summary: KCa3.1阻断剂
      ≥17.25 mg/mL
      insoluble in H2O
  7. Teneligliptin hydrobromide
    A3865 Teneligliptin hydrobromide
    中文名: 氢溴酸替格列汀
    Target: DPP-4
    Summary: DDP4抑制剂
      ≥62.9 mg/mL
      ≥104.8 mg/mL
  8. Phloretin
    A3723 Phloretin
    中文名: 根皮素
    Target: SGLT
    Summary: 在苹果中发现的二氢查耳酮
      ≥105 mg/mL
      insoluble in H2O
  9. Alogliptin (SYR-322)
    A4038 Alogliptin (SYR-322)
     1 Citation
    中文名: 阿格列汀
    Target: DPP-4
    Summary: DPP-4抑制剂
      ≥14.75 mg/mL
      insoluble in H2O
  10. Sitagliptin phosphate monohydrate
    A4036 Sitagliptin phosphate monohydrate
     5 Citation
    中文名: 磷酸西他列汀一水合物
    Target: DPP-4
    Summary: DPP-4抑制剂
      ≥23.8 mg/mL
      ≥30.6 mg/mL

10 件产品

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