Signaling Pathways - Protease-Activated Receptors - Hypoxia-Inducible Factor Prolyl Hydroxylase Inhibitors (HIF-PHIs) - p53
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- A8809 Vorapaxar中文名: 沃拉帕沙Target: Protease-Activated ReceptorsSummary: PAR-1拮抗剂
- A8229 ML161Target: Protease-Activated ReceptorsSummary: PAR1抑制剂
- A4482 Pifithrin-μ1 CitationTarget: Autophagy|p53|HSP70Summary: p53结合抑制剂,抗凋亡。
- A4506 DMOGTarget: Hypoxia-Inducible Factor Prolyl Hydroxylase Inhibitors (HIF-PHIs)Summary: 细胞通透的竞争性HIF-PH抑制剂
- A4483 PRIMA-1Target: p53Summary: BAX抑制剂
- A4481 PhiKan 083Target: p53Summary: P53稳定剂
- A4203 Tenovin-1Target: Sir2-like Family Deacetylases (Sirtuins)|p53|p21Summary: SIRT2 抑制剂,p53激活剂
- A4204 JNJ-26854165 (Serdemetan)1 CitationTarget: p53|HDM2 ubiquitin ligaseSummary: P53激活剂,阻断Mdm2-p53相互作用。
- A4206 Pifithrin-α (PFTα)2 CitationTarget: p53Summary: p53抑制剂
- A4208 NSC 319726Target: p53Summary: 突变型p53的活性剂