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Signaling Pathways - Aminopeptidases - PKA - Serotonin reuptake - Adenosine A2A Receptors

18件产品中的 1-10

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  1. Regadenoson
    B5904 Regadenoson
     1 Citation
    中文名: 类伽腺苷
    Target: Adenosine A2A Receptors
    Summary: A2A腺苷受体激动剂
      ≥18.05 mg/mL
      insoluble in H2O
  2. SCH 58261
    B6995 SCH 58261
    Target: Adenosine A2A Receptors
    Summary: A2A腺苷受体竞争性拮抗剂
      ≥34.5 mg/mL
      insoluble in H2O
  3. H-7 dihydrochloride
    B6342 H-7 dihydrochloride
    Target: PKC|PKG|PKA|Myosin light chain kinases (MLCKs)
    Summary: 蛋白激酶抑制剂
      Soluble in DMSO
  4. Midostaurin (PKC412)
    B3709 Midostaurin (PKC412)
    中文名: 米哚妥林
    Target: PKC|PKA|KDR|Flk1|PPK|c-Syk|CDK1/CyclinB
    Summary: PKC抑制剂
      ≥57.1 mg/mL
      insoluble in H2O
  5. 8-Bromo-cAMP, sodium salt
    B9000 8-Bromo-cAMP, sodium salt
    中文名: 8-溴腺苷3',5'-环腺苷一磷酸
    Target: PKA
    Summary: 细胞渗透性cAMP类似物,激活PKA
      ≥22.43 mg/mL
      ≥43 mg/mL
  6. Fasudil
    B3523 Fasudil
    中文名: 法舒地尔
    Target: ROCK|PKC|PKG|PKA|Myosin light chain kinases (MLCKs)
    Summary: 钙拮抗剂
      Soluble in DMSO
  7. Fluvoxamine
    B1205 Fluvoxamine
    中文名: 氟伏沙明
    Target: Serotonin reuptake
    Summary: 选择性5-羟色胺再摄取抑制剂
      ≥15.92 mg/mL
      insoluble in H2O
  8. Bestatin hydrochloride
    A8621 Bestatin hydrochloride
    中文名: 盐酸乌苯美司
    Target: Aminopeptidases
    Summary: 氨肽酶N(APN/CD13)和氨肽酶B抑制剂。
      ≥125 mg/mL
      ≥34.2 mg/mL
  9. A-674563
    A8616 A-674563
    Target: Cyclin-Dependent Kinases|Akt|GSK-3|ERK|PKC|PKA|RSK
    Summary: Akt1 / PKA / CDK2的强效选择性抑制剂
      ≥4.9 mg/mL
      ≥23.8 mg/mL
  10. Istradefylline (KW-6002)
    A8454 Istradefylline (KW-6002)
    中文名: 伊曲茶碱
    Target: Adenosine A2A Receptors
    Summary: 选择性A2A受体拮抗剂
      ≥8.78 mg/mL
      insoluble in H2O

18件产品中的 1-10

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