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Signaling Pathways - Histone Demethylases - Cytochrome P450 (CYP450) - GSK-3 - Cancer

11件产品中的 1-10

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  1. SP2509
    B4894 SP2509
    Target: Histone Demethylases
    Summary: 新型LSD1拮抗剂
      ≥19.45 mg/mL
      insoluble in H2O
  2. Indirubin
    B3672 Indirubin
    中文名: 靛玉红
    Target: Cyclin-Dependent Kinases|GSK-3
    Summary: 细胞周期蛋白依赖性激酶和GSK-3β抑制剂
      ≥13.1 mg/mL
      insoluble in H2O
  3. TOK-001
    A8623 TOK-001
    中文名: 加来特龙,伽来特隆
    Target: Androgen Receptors|Cytochrome P450 (CYP450)
    Summary: CYP17抑制剂和雄激素受体(AR)拮抗剂
      ≥12.4 mg/mL
      insoluble in H2O
  4. A-674563
    A8616 A-674563
    Target: Cyclin-Dependent Kinases|Akt|GSK-3|ERK|PKC|PKA|RSK
    Summary: Akt1 / PKA / CDK2的强效选择性抑制剂
      ≥4.9 mg/mL
      ≥23.8 mg/mL
  5. Thioridazine HCl
    A8537 Thioridazine HCl
    中文名: 盐酸硫利达嗪,盐酸硫代利哒,甲硫达嗪盐酸盐,甲硫哒嗪盐酸盐
    Target: Cytochrome P450 (CYP450)|D1 and D5 Receptors|D2 Receptors|D3 Receptors|D4 Receptors
    Summary: 钙通道蛋白抑制剂
      ≥20.35 mg/mL
      ≥6.78 mg/mL
  6. Zosuquidar
    A3956 Zosuquidar
    Target: P-glycoprotein (P-gp)|Cytochrome P450 (CYP450)
    Summary: MDR调节剂
      Soluble in DMSO
  7. LY2090314
    A3570 LY2090314
    Target: GSK-3
    Summary: 有效的GSK-3抑制剂
      ≥91 mg/mL
      insoluble in H2O
  8. AR-A014418
    A3184 AR-A014418
     2 Citation
    Target: GSK-3
    Summary: GSK3β抑制剂
      ≥15.4 mg/mL
      insoluble in H2O
  9. Ketoconazole
    A4316 Ketoconazole
    中文名: 酮康唑
    Target: Cytochrome P450 (CYP450)
    Summary: 环孢菌素氧化酶和睾酮6β-羟化酶的抑制剂
      ≥23.4 mg/mL
      insoluble in H2O
  10. Abiraterone acetate
    A8202 Abiraterone acetate
    中文名: 乙酸阿比特龙酯
    Target: Cytochrome P450 (CYP450)
    Summary: 细胞色素p450 17a1抑制剂
      ≥11.22 mg/mL
      insoluble in H2O

11件产品中的 1-10

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