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Signaling Pathways - Histone Demethylases - Cytochrome P450 (CYP450) - Caspases - Cancer

10 件产品

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  1. SP2509
    B4894 SP2509
    Target: Histone Demethylases
    Summary: 新型LSD1拮抗剂
      ≥19.45 mg/mL
      insoluble in H2O
  2. Z-IETD-FMK
    B3232 Z-IETD-FMK
     12 Citation
    Target: Caspases
    Summary: Caspase-8抑制剂
      ≥32.73 mg/mL
      insoluble in H2O
  3. TOK-001
    A8623 TOK-001
    中文名: 加来特龙,伽来特隆
    Target: Androgen Receptors|Cytochrome P450 (CYP450)
    Summary: CYP17抑制剂和雄激素受体(AR)拮抗剂
      ≥12.4 mg/mL
      insoluble in H2O
  4. Thioridazine HCl
    A8537 Thioridazine HCl
    中文名: 盐酸硫利达嗪,盐酸硫代利哒,甲硫达嗪盐酸盐,甲硫哒嗪盐酸盐
    Target: Cytochrome P450 (CYP450)|D1 and D5 Receptors|D2 Receptors|D3 Receptors|D4 Receptors
    Summary: 钙通道蛋白抑制剂
      ≥20.35 mg/mL
      ≥6.78 mg/mL
  5. Zosuquidar
    A3956 Zosuquidar
    Target: P-glycoprotein (P-gp)|Cytochrome P450 (CYP450)
    Summary: MDR调节剂
      Soluble in DMSO
  6. Z-DQMD-FMK
    A1921 Z-DQMD-FMK
     3 Citation
    Target: Caspases
    Summary: 细胞渗透性Caspase-3抑制剂
      ≥29.2 mg/mL
      insoluble in H2O
  7. Ketoconazole
    A4316 Ketoconazole
    中文名: 酮康唑
    Target: Cytochrome P450 (CYP450)
    Summary: 环孢菌素氧化酶和睾酮6β-羟化酶的抑制剂
      ≥23.4 mg/mL
      insoluble in H2O
  8. Q-VD-OPh
    A1901 Q-VD-OPh
     53 Citation
    Target: Caspases
    Summary: Pan-caspase抑制剂。
      ≥25.67 mg/mL
      insoluble in H2O
  9. Abiraterone acetate
    A8202 Abiraterone acetate
    中文名: 乙酸阿比特龙酯
    Target: Cytochrome P450 (CYP450)
    Summary: 细胞色素p450 17a1抑制剂
      ≥11.22 mg/mL
      insoluble in H2O
  10. PAC-1
    A8177 PAC-1
     1 Citation
    Target: Caspases
    Summary: 半胱天冬酶-3酶原激活剂
      ≥13.4 mg/mL
      insoluble in H2O

10 件产品

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