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Signaling Pathways - MST - Ron - Inositol-requiring enzyme 1 (IRE1) - Src

22件产品中的 11-20

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  1. Butein
    A2689 Butein
    中文名: 紫铆因,紫铆查尔酮
    Target: Src|STAT|EGFR|Angiotensin-Converting Enzymes (ACEs)|5-Lipoxygenases|PTK|enoyl-acyl-carrier protein reductase
    Summary: 蛋白激酶抑制剂
      ≥13.6 mg/mL
      insoluble in H2O
  2. Ponatinib (AP24534)
    A5467 Ponatinib (AP24534)
     1 Citation
    中文名: 帕纳替尼
    Target: VEGFR|PDGFR|Bcr-Abl|FGFR|Src
    Summary: pan-BCR-ABL抑制剂,多激酶抑制剂
      ≥53.3 mg/mL
      insoluble in H2O
  3. Saracatinib (AZD0530)
    A2133 Saracatinib (AZD0530)
     3 Citation
    中文名: 塞卡替尼
    Target: Src
    Summary: Src/Abl抑制剂
      ≥27.1 mg/mL
      ≥2.36 mg/mL
  4. CP-724714
    A2412 CP-724714
    Target: VEGFR|PDGFR|Bcr-Abl|Src|EGFR|c-MET|Insulin Receptors|IRG-1R
    Summary: 有效的HER2选择性抑制剂
      ≥23.5 mg/mL
      insoluble in H2O
  5. Bosutinib (SKI-606)
    A2149 Bosutinib (SKI-606)
     1 Citation
    中文名: 伯舒替尼
    Target: Bcr-Abl|Src
    Summary: Abl/Src有效的抑制剂
      ≥26.5 mg/mL
      insoluble in H2O
  6. PP 1
    A8215 PP 1
    Target: Src|EGFR|JAK|ZAP-70
    Summary: Src家族酪氨酸激酶抑制剂
      ≥7.03 mg/mL
      insoluble in H2O
  7. TG 100801
    A3870 TG 100801
    Target: VEGFR|FGFR|Src|Fyn kinase
    Summary: 多激酶抑制剂
      Soluble in DMSO
  8. KX2-391 dihydrochloride
    A3535 KX2-391 dihydrochloride
    Target: Src
    Summary: Src激酶抑制剂
      ≥25.2 mg/mL
      insoluble in H2O
  9. TAK-901
    A4124 TAK-901
    Target: Aurora Kinases|FLT3|Src|JAK|LRRK2|Hck|FGR|YES|Fyn|ARG
    Summary: Aurora A/B抑制剂
      ≥25.25 mg/mL
      insoluble in H2O
  10. ENMD-2076
    A4130 ENMD-2076
    Target: Aurora Kinases|FLT3|RET|Src|VEGFR3/FLT4|NTRK1/TRKA|CSF-1R/c-Fms
    Summary: Aurora A/Flt3的选择性抑制剂
      ≥18.75 mg/mL
      insoluble in H2O

22件产品中的 11-20

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