切换导航
关闭
  • 菜单
  • Setting

Signaling Pathways - Sphingosine kinases (SphKs) - BCPCF efflux - Cytochrome P450 (CYP450) - CFTR

22件产品中的 11-20

页面
每页
清除全部
  1. Clotrimazole
    A8401 Clotrimazole
     2 Citation
    中文名: 克霉唑
    Target: Cytochrome P450 (CYP450)
    Summary: 抗真菌化合物
      ≥28.1 mg/mL
      insoluble in H2O
  2. Thioridazine HCl
    A8537 Thioridazine HCl
    中文名: 盐酸硫利达嗪,盐酸硫代利哒,甲硫达嗪盐酸盐,甲硫哒嗪盐酸盐
    Target: Cytochrome P450 (CYP450)|D1 and D5 Receptors|D2 Receptors|D3 Receptors|D4 Receptors
    Summary: 钙通道蛋白抑制剂
      ≥20.35 mg/mL
      ≥6.78 mg/mL
  3. VX-809
    A8351 VX-809
    中文名: 鲁玛卡托
    Target: CFTR
    Summary: CFTR调节剂
      ≥22.6 mg/mL
      insoluble in H2O
  4. VX-661
    A2664 VX-661
    Target: CFTR
    Summary: F508del CFTR校正子
      ≥21.8 mg/mL
      ≥24.3 mg/mL
  5. Posaconazole
    A1718 Posaconazole
    中文名: 泊沙康唑
    Target: Cytochrome P450 (CYP450)|sterol demethylase
    Summary: 甾醇 C14ɑ去甲基化酶抑制剂
      ≥35.04 mg/mL
      insoluble in H2O
  6. Zosuquidar
    A3956 Zosuquidar
    Target: P-glycoprotein (P-gp)|Cytochrome P450 (CYP450)
    Summary: MDR调节剂
      Soluble in DMSO
  7. PF-543
    A3717 PF-543
     1 Citation
    Target: Sphingosine kinases (SphKs)
    Summary: SphK1选择性抑制剂
      ≥23.3 mg/mL
      insoluble in H2O
  8. Dronedarone
    A3374 Dronedarone
    中文名: 决奈达隆
    Target: Cytochrome P450 (CYP450)|sodium channel|adrenergic receptor|potassium channel|calcium channel
    Summary: CYP3A4和2D6抑制剂
      ≥27.84 mg/mL
      insoluble in H2O
  9. Clarithromycin
    A4322 Clarithromycin
    中文名: 克拉霉素
    Target: Cytochrome P450 (CYP450)
    Summary: CYP3A抑制剂
      ≥31.2 mg/mL
      insoluble in H2O
  10. Ketoconazole
    A4316 Ketoconazole
    中文名: 酮康唑
    Target: Cytochrome P450 (CYP450)
    Summary: 环孢菌素氧化酶和睾酮6β-羟化酶的抑制剂
      ≥23.4 mg/mL
      insoluble in H2O

22件产品中的 11-20

页面
每页