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- A1910 Bromodomain Inhibitor, (+)-JQ138 CitationTarget: BromodomainsSummary: BET bromodomain抑制剂。
- A2942 Masitinib (AB1010)中文名: 马赛替尼Target: PDGFR|c-Kit|LynSummary: 酪氨酸激酶抑制剂
- B5839 SU6656Target: Src|Lyn|YES|FynSummary: Src 酪氨酸激酶抑制剂
- B7675 DIDSTarget: voltage-gated chloride channelsSummary: 阴离子运输抑制剂
- B1012 MS436Target: BromodomainsSummary: BRD4抑制剂
- A4186 Bromosporine1 CitationTarget: BromodomainsSummary: Bromodomain抑制剂
- B1498 I-BET-7624 CitationTarget: BromodomainsSummary: BET抑制剂
- A4184 PFI-1 (PF-6405761)1 CitationTarget: BromodomainsSummary: BET抑制剂
- B1013 GSK1324726ATarget: BromodomainsSummary: BET蛋白抑制剂
- A3692 OTX-0153 Citation中文名: 比拉瑞塞Target: BromodomainsSummary: BRD抑制剂