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- A1910 Bromodomain Inhibitor, (+)-JQ138 CitationTarget: BromodomainsSummary: BET bromodomain抑制剂。
- A8218 Lapatinib2 Citation中文名: 拉帕替尼Target: ErbBSummary: EGFR/HER2抑制剂
- A4092 CUDC-1011 CitationTarget: Histone Deacetylases (HDACs)|EGFR|ErbBSummary: 多靶点HDAC抑制剂
- A8319 Dacomitinib (PF299804, PF299)中文名: 达克替尼Target: ErbBSummary: HER抑制剂
- A8375 AZD8931 (Sapitinib)中文名: 沙普替尼Target: EGFR|ErbBSummary: ErbB抑制剂
- B7675 DIDSTarget: voltage-gated chloride channelsSummary: 阴离子运输抑制剂
- B1012 MS436Target: BromodomainsSummary: BRD4抑制剂
- B1543 Mubritinib (TAK 165)中文名: 木利替尼Target: ErbBSummary: HER2/ErbB2有效抑制剂
- A4186 Bromosporine1 CitationTarget: BromodomainsSummary: Bromodomain抑制剂
- B1498 I-BET-7624 CitationTarget: BromodomainsSummary: BET抑制剂