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- A8215 PP 1Target: Src|EGFR|JAK|ZAP-70Summary: Src家族酪氨酸激酶抑制剂
- A4166 EPZ56761 CitationTarget: DOT1LSummary: DOT1L抑制剂
- A3543 LDE225 DiphosphateTarget: SmoothenedSummary: Smo拮抗剂
- A5703 BMS-777607Target: METSummary: 强效的c-Met选择性抑制剂
- A3010 MK-2206 dihydrochloride21 CitationTarget: AktSummary: Akt1/2/3抑制剂
- A8171 Entinostat (MS-275,SNDX-275)2 Citation中文名: 恩替诺特Target: Histone Deacetylases (HDACs)Summary: HDAC1和HDAC3抑制剂
- N2791 Cucurbitacin E中文名: 葫芦素 ETarget: ActinSummary: 抑制肌动蛋白解聚
- B7070 Triacsin CTarget: Synthases/SynthetasesSummary: 酰基辅酶A合成酶抑制剂
- N1375 Solamargine中文名: 澳洲茄边碱,边缘茄碱Summary: 细胞毒性剂
- B7207 SecinH3Target: Guanine nucleotide exchange factors (GEFs)Summary: Sec7特异性GEF抑制剂