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- B1236 BML-277Target: ChkSummary: 有效的Chk2选择性抑制剂
- B1964 Lonidamine中文名: 氯尼达明Target: HexokinasesSummary: 己糖激酶失活剂
- B5880 CCT244747Target: ChkSummary: CHK1抑制剂
- B1232 XL413Target: Cdc7Summary: Cdc7抑制剂
- A3721 PHA-767491Target: Cyclin-Dependent Kinases|MK2|Cdc7Summary: Cdc7 / CDK9抑制剂
- B1088 LY2606368Target: ChkSummary: CHK1抑制剂
- B1437 PF-477736Target: ChkSummary: Chk1抑制剂
- A3291 CCT241533Target: ChkSummary: 有效的Chk2抑制剂
- A5919 AZD7762Target: ChkSummary: ATP竞争性的检查点激酶抑制剂
- A8394 CHIR-124Target: FLT3|GSK-3|Chk|PDGFRSummary: Chk1抑制剂