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- B2172 PP121Target: mTOR|Eph Receptors|VEGFR|PDGFR|Bcr-Abl|Src|DNA-PK|P110|HckSummary: 酪氨酸激酶和磷酸肌醇激酶双重抑制剂
- A2949 Linifanib (ABT-869)Target: VEGFR|PDGFRSummary: VEGFR/PDGFR抑制剂
- B6431 Zinc protoporphyrin IX2 Citation中文名: 锌原卟啉Target: Guanylyl Cyclases|Heme oxygenaseSummary: 血红素加氧酶抑制剂
- B7354 SU 16fTarget: PDGFRSummary: PDGFRβ抑制剂
- N1842 Taxifolin中文名: 紫杉叶素,黄杉素Target: AdipoR2|Opioid receptors
- B7641 YC 1中文名: 利非西呱Target: Guanylyl CyclasesSummary: 可溶性鸟苷酸环化酶(sGC)激活剂
- A2174 Lenvatinib (E7080)中文名: 乐伐替尼,仑伐替尼Target: VEGFR|PDGFR|RETSummary: VEGFR抑制剂
- B5835 AZD2932Target: FLT3|VEGFR|PDGFR|c-KitSummary: VEGFR-2\PDGFRβ\Flt-3和c-Kit的抑制剂
- A8550 Telatinib (BAY 57-9352)中文名: 替拉替尼Target: VEGFR|PDGFR|c-KitSummary: VEGFR-2/-3、PDGFR-β和c-Kit抑制剂
- B1879 AdipoRonTarget: AdipoR1|AdipoR2Summary: AdipoR1/2激动剂