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- A8704 Stiripentol中文名: 司替戊醇Target: Lactate Dehydrogenases (LDH)Summary: LDH抑制剂
- A5354 Zonisamide中文名: 唑尼沙胺Target: Voltage-gated Sodium (NaV) Channels|Voltage-gated Calcium Channels (CaV)|Carbonic Anhydrases|Calcium-Activated Potassium (KCa) ChannelsSummary: 抗惊厥和机械效应的抗癫痫药
- A8332 R788 disodium中文名: 福他替尼二钠盐Target: SykSummary: Syk的ATP竞争性抑制剂
- A4317 Apremilast (CC-10004)中文名: 阿普斯特Target: Phosphodiesterases (PDEs)Summary: PDE4抑制剂
- A5176 AS-605240Target: PI3KSummary: PI 3-Kγ选择性抑制剂
- B1642 WYE-125132 (WYE-132)Target: mTORSummary: mTOR抑制剂
- A1987 Ki164254 CitationTarget: LPA ReceptorsSummary: LPA受体拮抗剂
- A1198 Levetiracetam中文名: 左乙拉西坦Summary: 抗癫痫药物
- B2284 Fostamatinib (R788)中文名: 福坦替尼Target: SykSummary: 脾酪氨酸激酶(Syk)抑制剂
- A3284 Cathepsin S inhibitor1 CitationTarget: CathepsinsSummary: 抑制MHCII抗原呈递