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- B6988 BRL 50481Target: Phosphodiesterases (PDEs)Summary: PDE7抑制剂
- B2186 GSK2636771Target: PI3KSummary: PIK3抑制剂
- A3209 AXL1717中文名: 鬼臼毒素Target: Insulin-like growth factor receptors(IGFRs)Summary: IGF-1R抑制剂,口服有效。
- A1877 XAV-9391 CitationTarget: TNKSSummary: Tankyrase 1/2抑制剂
- B1642 WYE-125132 (WYE-132)Target: mTORSummary: mTOR抑制剂
- A3721 PHA-767491Target: Cyclin-Dependent Kinases|MK2|Cdc7Summary: Cdc7 / CDK9抑制剂
- A1987 Ki164254 CitationTarget: LPA ReceptorsSummary: LPA受体拮抗剂
- A4010 Salinosporamide A (NPI-0052, Marizomib)Target: ProteasomeSummary: 20S蛋白酶体抑制剂
- B2173 CP-673451Target: PDGFRSummary: PDGFRα/β抑制剂
- B1772 Ibandronate sodium中文名: 伊班膦酸钠一水合物Target: Bone resorptionSummary: 双膦酸盐药物