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- B2186 GSK2636771Target: PI3KSummary: PIK3抑制剂
- B6988 BRL 50481Target: Phosphodiesterases (PDEs)Summary: PDE7抑制剂
- A1196 SGX-5231 CitationTarget: METSummary: 高度选择性的、ATP竞争性的Met抑制剂
- B2173 CP-673451Target: PDGFRSummary: PDGFRα/β抑制剂
- A1821 Ki8751Target: VEGFRSummary: VEGFR-2有效的、选择性抑制剂
- A3712 PF-04217903 methanesulfonateTarget: c-METSummary: c-Met抑制剂
- A3573 LY2801653Target: METSummary: MET抑制剂
- B1772 Ibandronate sodium中文名: 伊班膦酸钠一水合物Target: Bone resorptionSummary: 双膦酸盐药物
- A4365 Lovastatin中文名: 洛伐他汀Target: HMG-CoA ReductasesSummary: HMG-CoA还原酶抑制剂
- A1915 Zebularine1 Citation中文名: 泽布拉林Target: DNA Methyltransferases|Cytidine deaminasesSummary: DNA甲基化抑制剂