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- B5421 (Z)-4-Hydroxytamoxifen中文名: 4-羟基他莫昔芬Target: Estrogen and Related ReceptorsSummary: 雌激素受体(ER)调节剂
- A3632 Motesanib中文名: 莫特塞尼Target: VEGFRSummary: Flk-1/Flt-4/PDGFR-/c-Kit抑制剂
- A3412 Fenretinide中文名: 维甲酰酚胺Target: FAKSummary: 合成的维甲酸激动剂
- A4393 Paclitaxel (Taxol)4 Citation中文名: 紫杉醇Target: Microtubules/TubulinsSummary: 抗肿瘤药
- B3941 Talabostat mesylate2 CitationTarget: DPP-4Summary: DPP4抑制剂
- A8353 3-Methyladenine3 Citation中文名: 3-甲基腺嘌呤Target: PI3KSummary: III类PI3K抑制剂
- A4083 Rocilinostat (ACY-1215)1 CitationTarget: Histone Deacetylases (HDACs)Summary: 选择性的HDAC6抑制剂
- A8208 Tariquidar2 Citation中文名: 他立喹达Target: P-glycoprotein (P-gp)Summary: P-糖蛋白抑制剂
- A4097 CUDC-907中文名: 非美诺司他Target: Histone Deacetylases (HDACs)|PI3KSummary: PI3K/HDAC抑制剂
- A3818 SilvestrolSummary: 抗肿瘤药