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- A8351 VX-809中文名: 鲁玛卡托Target: CFTRSummary: CFTR调节剂
- A4335 Mildronate中文名: 米屈肼Target: Hydroxylases|carnitine reabsorptionSummary: GBB羟化酶抑制剂
- A8637 IOWH-032Target: CFTRSummary: CFTR抑制剂
- A8476 MK-2461Target: FLT3|PDGFR|MET|RonSummary: C-Met(野生型/突变型)抑制剂
- B2087 Ciclopirox中文名: 环吡酮胺Target: HydroxylasesSummary: 广谱抗真菌剂
- B4751 L-MimosineTarget: HydroxylasesSummary: 铁螯合剂和脯氨酰-4-羟化酶抑制剂
- B1087 GlyH-101Target: CFTRSummary: CFTR Inhibitor II
- A2664 VX-661Target: CFTRSummary: F508del CFTR校正子