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- B1640 Torin 21 CitationTarget: mTOR|DNA-PK|ATM/ATRSummary: MTOR抑制剂
- A2412 CP-724714Target: VEGFR|PDGFR|Bcr-Abl|Src|EGFR|c-MET|Insulin Receptors|IRG-1RSummary: 有效的HER2选择性抑制剂
- A8336 KU-600192 CitationTarget: ATM/ATRSummary: ATM激酶抑制剂
- A8624 CGK733Target: ATM/ATRSummary: ATM/ATR抑制剂
- A3173 AMD-070Target: CXCRSummary: CXCR4拮抗剂
- B3266 AMG 4871 CitationTarget: CXCRSummary: CXCR3拮抗剂
- A3753 Reparixin L-lysine salt1 Citation中文名: 瑞帕利辛L-赖氨酸盐Target: CXCRSummary: CXCL8受体CXCR1/CXCR2活化的抑制剂
- A3803 SCH 563705Target: CXCRSummary: CXCR2/CXCR1拮抗剂
- B6007 AZD67381 CitationTarget: ATM/ATRSummary: ATR抑制剂
- A1986 Nu 6027Target: Cyclin-Dependent Kinases|ATM/ATRSummary: 有效的ATR/CDK选择性抑制剂