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- A4132 CCT137690Target: Aurora KinasesSummary: Aurora A / B / C抑制剂
- B1104 AZD-92911 Citation中文名: 奥希替尼Target: EGFRSummary: 突变型EGFR抑制剂。
- A8487 Nocodazole1 Citation中文名: 诺考达唑Target: Microtubules/TubulinsSummary: 微管蛋白产生抑制剂,抗肿瘤剂
- A1769 KU-00606481 CitationTarget: PI3K|DNA-PKSummary: DNA-PK/PI3-K双重抑制剂
- A3004 Vemurafenib (PLX4032, RG7204)9 Citation中文名: 维罗非尼Target: RafSummary: BRAF激酶抑制剂
- A3692 OTX-0153 Citation中文名: 比拉瑞塞Target: BromodomainsSummary: BRD抑制剂
- B1288 RigosertibTarget: PI3K|PLKSummary: PI3K/PLK1抑制剂
- B2186 GSK2636771Target: PI3KSummary: PIK3抑制剂
- B6342 H-7 dihydrochlorideTarget: PKC|PKG|PKA|Myosin light chain kinases (MLCKs)Summary: 蛋白激酶抑制剂
- A4413 PD 150606Target: CalpainsSummary: 非肽类钙蛋白酶抑制剂