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- A4326 TAK-700 (Orteronel)2 CitationTarget: human lyaseSummary: 人17,20-裂解酶抑制剂
- N1656 Schizandrin B中文名: 五味子醇乙Target: Nrf2|ROS and Other Gaseous DonorsSummary: 抑制脂质过氧化
- A8218 Lapatinib2 Citation中文名: 拉帕替尼Target: ErbBSummary: EGFR/HER2抑制剂
- B7795 Toyocamycin中文名: 丰加霉素Target: phosphatidylinositol kinaseSummary: 腺苷类似物,抗肿瘤抗生素
- A4092 CUDC-1011 CitationTarget: Histone Deacetylases (HDACs)|EGFR|ErbBSummary: 多靶点HDAC抑制剂
- B1543 Mubritinib (TAK 165)中文名: 木利替尼Target: ErbBSummary: HER2/ErbB2有效抑制剂
- A8375 AZD8931 (Sapitinib)中文名: 沙普替尼Target: EGFR|ErbBSummary: ErbB抑制剂