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- A1020 GnRH Associated Peptide (1-13), humanTarget: prolactin secretion|gonadotropin releaseSummary: 催乳素分泌抑制剂
- B1437 PF-477736Target: ChkSummary: Chk1抑制剂
- A8477 MK-8776 (SCH-900776)Target: ChkSummary: Chk1高效选择性抑制剂
- A8621 Bestatin hydrochloride中文名: 盐酸乌苯美司Target: AminopeptidasesSummary: 氨肽酶N(APN/CD13)和氨肽酶B抑制剂。
- A3291 CCT241533Target: ChkSummary: 有效的Chk2抑制剂
- N1359 Magnolol中文名: 厚朴酚Target: CB1 Receptors|NO Donors / Precursors|CB2 ReceptorsSummary: NO/TNF-α产生的抑制剂;抗真菌剂
- A5919 AZD7762Target: ChkSummary: ATP竞争性的检查点激酶抑制剂
- A3850 TAK-2427 Citation中文名: 瑞沙托维Target: Toll-like receptors (TLRs)|NO Donors / Precursors|IL ReceptorsSummary: TLR 4信号抑制剂
- B1236 BML-277Target: ChkSummary: 有效的Chk2选择性抑制剂
- A3237 Betulinic acid中文名: 白桦脂酸,桦木酸Target: Aminopeptidases|Topoisomerases|HIVSummary: 抗HIV和抗肿瘤化合物,五环三萜类化合物